Clinical Pharmacology Details


Mesterolone


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Indications & Dose:

Adults:


Potency disturbances:   



Initially, 25mg (1 tab) thrice daily till satisfactory response achieved. .


Maint dose: 25mg (1 tab) 1-2 times daily.


Hypogonadism:



25-50mg (1-2 tabs) thrice daily for several months.


Maint: 25mg (1 tab) 2-3 times daily.


Male infertility:  



25mg (1 tab) 2-3 times daily for a cycle of spermatogenesis i.e. about 90 days.

Contraindications:

Carcinoma of prostate, carcinoma of liver. Females. Pregnancy & breastfeeding: 

Side Effects:

 Frequent erection, priapism. 

Cautions:

Precautions:

Prostate to be examined prophylactically. For use in male patients only.
Old age: May be used. 

Interaction:

Drugs
See under androgens. 

Warnings:

Adverse Effects:

Lactations:

Special Precautions:

Counselling:

Side Effects Or Adverse Reactions:

Patient And Carer Advice: