Clinical Pharmacology Details


FLUTICASONE


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Indications & Dose:

Prophylaxis of asthma



Child 5–15 years: Initially 50–100 micrograms twice daily (max. per dose 200 micrograms twice daily), dose to be adjusted as necessary


Child 16–17 years: Initially 100–500 micrograms twice daily (max. per dose 1 mg twice daily), dose may be increased according to severity of asthma. Doses above 500 micrograms twice daily initiated by aspecialist


Adult: Initially 100–500 micrograms twice daily (max. per dose 1 mg twice daily), dose may be increased according to severity of asthma. Doses above 500 micrograms twice daily initiated by a specialist



Child 4–15 years: Initially 50–100 micrograms twice daily (max. per dose 200 micrograms twice daily), dose to be adjusted as necessary


Child 16–17 years: Initially 100–500 micrograms twice daily (max. per dose 1 mg twice daily), dose may be increased according to severity of asthma. Doses above 500 micrograms twice daily initiated by a specialist Adult: Initially 100–500 micrograms twice daily (max. per dose 1 mg twice daily), dose may be increased according to severity of asthma. Doses above 500 micrograms twice daily initiated by a specialist



Child 4–15 years: 1 mg twice daily


Child 16–17 years: 0.5–2 mg twice daily


Adult: 0.5–2 mg twice daily 


 

Contraindications:

Relief of acute bronchospasm


PREGNANCY AND LACTATION: Pregnancy category Q no information on excretion into human breast milk 

Side Effects:

CNS: Fatigue, headache


EENT: Dysphonia, nasal congestion or discharge, oropharyngeal candidiasis, sinusitis, upper respiratory tract infections


VS: Muscle soreness


RESP: Bronchospasm


SKIN.. Urticaria


MISC: Angioedema, hypersensitivity reactions (shortness of breath, tightness in chest, wheezing)

Cautions:

Precautions:

Interaction:

Drugs


• Ketoconazole: Possible increased plasma fluticasone concentrations 

Warnings:

Adverse Effects:

Lactations:

Special Precautions:

Counselling:

Side Effects Or Adverse Reactions:

Patient And Carer Advice: